留可然有什么特点?


留可然的治疗作用有哪些特点?

  你好!留可然(苯丁酸氮芥片)属氮芥类衍生物,具有双功能烷化剂作用,可形成不稳定的乙撑亚胺而发挥其细胞毒作用,干扰DNA和RNA的功能。在常规剂量下,其毒性较其他任何氮芥类药物小。对增殖状态的细胞敏感,特别对G1期与M期的作用最强,属细胞周期非特异性药物。对了霍奇金病,数种非霍奇金病淋巴瘤,慢性淋巴细胞性白血病,瓦尔登斯特伦巨球蛋白血症,晚期卵巢腺癌。留可然对于部分乳腺癌病人也有明显的疗效。对淋巴细胞癌也有一定的选择性控制作用。
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